• 咨询热线
    客服服务热线 13671568941/15317326293
  • 在线咨询
  • 微信客服
    微信客服
  • 公众号
    扫码关注公众号

Eg5 Inhibitor V, trans-24

CAS No. 869304-55-2

Eg5 Inhibitor V, trans-24 ( —— )

产品货号. M26190 CAS No. 869304-55-2

Eg5 Inhibitor V, trans-24 is a specific and potent Eg5 agonist inhibitor that can be used in cancer research with an IC50 value of 0.65 uM.

纯度: >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
规格 价格/人民币 库存 数量
2MG ¥1887 有现货
5MG ¥2900 有现货
10MG ¥4342 有现货
25MG ¥7023 有现货
50MG ¥9639 有现货
100MG ¥12879 有现货
200MG 获取报价 有现货
500MG 获取报价 有现货
1G 获取报价 有现货

生物学信息

  • 产品名称
    Eg5 Inhibitor V, trans-24
  • 注意事项
    本公司产品仅用于科研实验,不得用于人体或动物的临床与诊断
  • 产品简述
    Eg5 Inhibitor V, trans-24 is a specific and potent Eg5 agonist inhibitor that can be used in cancer research with an IC50 value of 0.65 uM.
  • 产品描述
    Eg5 Inhibitor V, trans-24 is a specific and potent Eg5 agonist inhibitor that can be used in cancer research with an IC50 value of 0.65 uM.(In Vitro):Trans-24 is a potent EG5-specific inhibitor with an IC50 conversion rate of 0.65 M and can be used in cancer research.
  • 同义词
    ——
  • 通路
    Cytoskeleton/Cell Adhesion Molecules
  • 靶点
    Kinesin
  • 受体
    Dyrk pS421; Dyrk1B
  • 研究领域
    ——
  • 适应症
    ——

化学信息

  • CAS Number
    869304-55-2
  • 分子量
    423.5
  • 分子式
    C26H21N3O3
  • 纯度
    >98% (HPLC)
  • 溶解度
    ——
  • SMILES
    [H][C@@]12Cc3c([nH]c4ccccc34)[C@H](N1C(=O)N(Cc1ccccc1)C2=O)c1cccc(O)c1
  • 化学全称
    ——

运输与储存

  • 储存条件
    (-20℃)
  • 运输条件
    With Ice Pack
  • 稳定性
    ≥ 2 years

参考文献

1.Kettle JG, et al. Discovery and optimization of a novel series of Dyrk1B kinase inhibitors to explore a MEK resistance hypothesis. J Med Chem. 2015 Mar 26;58(6):2834-44.
产品手册
关联产品
  • KSP-IA

    A potent, specific, allosteric and cell-active inhibitor of KSP with IC50 of 11 nM; has no ihibitory activity toward other kinesins.

  • BRD 9876

    BRD 9876 is an ATP- and ADP-competitive Eg5 (kinesin-5) inhibitor with Ki of 4 nM.

  • WZ8040

    WZ8040 is a novel mutant-selective irreversible EGFRT790M inhibitor, does not inhibit ERBB2 phosphorylation (T798I).