Eg5 Inhibitor V, trans-24
CAS No. 869304-55-2
Eg5 Inhibitor V, trans-24 ( —— )
产品货号. M26190 CAS No. 869304-55-2
Eg5 Inhibitor V, trans-24 is a specific and potent Eg5 agonist inhibitor that can be used in cancer research with an IC50 value of 0.65 uM.
纯度: >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
规格 | 价格/人民币 | 库存 | 数量 |
2MG | ¥1887 | 有现货 |
|
5MG | ¥2900 | 有现货 |
|
10MG | ¥4342 | 有现货 |
|
25MG | ¥7023 | 有现货 |
|
50MG | ¥9639 | 有现货 |
|
100MG | ¥12879 | 有现货 |
|
200MG | 获取报价 | 有现货 |
|
500MG | 获取报价 | 有现货 |
|
1G | 获取报价 | 有现货 |
|
生物学信息
-
产品名称Eg5 Inhibitor V, trans-24
-
注意事项本公司产品仅用于科研实验,不得用于人体或动物的临床与诊断
-
产品简述Eg5 Inhibitor V, trans-24 is a specific and potent Eg5 agonist inhibitor that can be used in cancer research with an IC50 value of 0.65 uM.
-
产品描述Eg5 Inhibitor V, trans-24 is a specific and potent Eg5 agonist inhibitor that can be used in cancer research with an IC50 value of 0.65 uM.(In Vitro):Trans-24 is a potent EG5-specific inhibitor with an IC50 conversion rate of 0.65 M and can be used in cancer research.
-
同义词——
-
通路Cytoskeleton/Cell Adhesion Molecules
-
靶点Kinesin
-
受体Dyrk pS421; Dyrk1B
-
研究领域——
-
适应症——
化学信息
-
CAS Number869304-55-2
-
分子量423.5
-
分子式C26H21N3O3
-
纯度>98% (HPLC)
-
溶解度——
-
SMILES[H][C@@]12Cc3c([nH]c4ccccc34)[C@H](N1C(=O)N(Cc1ccccc1)C2=O)c1cccc(O)c1
-
化学全称——
运输与储存
-
储存条件(-20℃)
-
运输条件With Ice Pack
-
稳定性≥ 2 years
参考文献
1.Kettle JG, et al. Discovery and optimization of a novel series of Dyrk1B kinase inhibitors to explore a MEK resistance hypothesis. J Med Chem. 2015 Mar 26;58(6):2834-44.
产品手册
关联产品
-
KSP-IA
A potent, specific, allosteric and cell-active inhibitor of KSP with IC50 of 11 nM; has no ihibitory activity toward other kinesins.
-
BRD 9876
BRD 9876 is an ATP- and ADP-competitive Eg5 (kinesin-5) inhibitor with Ki of 4 nM.
-
WZ8040
WZ8040 is a novel mutant-selective irreversible EGFRT790M inhibitor, does not inhibit ERBB2 phosphorylation (T798I).